Compare
Catalogue No.
Description
GPCR Class
Target Sub-Family
Protein Target
Host Cells
HTS044M
ChemiScreen™ Membrane Preparation Human Recombinant M1 Muscarinic Acetylcholine Receptor
A
Acetylcholine (muscarinic)
M1
Chem-1
HTS115M
ChemiSCREEN™ Membrane Preparation Recombinant Human M2 Muscarinic Acetylcholine Receptor
A
Acetylcholine (muscarinic)
M2
Chem-1
HTS116M
ChemiSCREEN™ Human M3 Muscarinic Acetylcholine Receptor Membrane Preparation
A
Acetylcholine (muscarinic)
M3
Chem-1
HTS075M
ChemiScreen™ Membrane Preparation Recombinant Human M5 Muscarinic Acetylcholine Receptor
A
Acetylcholine (muscarinic)
M5
Chem-1
HTS047M
ChemiScreen™ A1 Membrane Preparation
A
Adenosine
A1
Chem-3
HTS052M
ChemiScreen™ A3 Membrane Preparation
A
Adenosine
A3
Chem-3
HTS087M
ChemiScreen™ Recombinant HumanMembrane Preparation α1A Adrenergic Receptor
A
Adrenergic
alpha1A
Chem-1
HTS158M
ChemiSCREEN™ Membrane Preparation Recombinant Human α1B Adrenergic Receptor
A
Adrenergic
alpha1B
Chem-1
HTS216M
ChemiSCREEN™ Membrane Preparation Recombinant Human α1D Adrenergic Receptor with N-terminal truncation
A
Adrenergic
alpha1D
Chem-1
HTS096M
ChemiSCREEN™ Human α2A Adrenergic Receptor Membrane Preparation
A
Adrenergic
alpha2A
Chem-1
HTS157M
ChemiSCREEN™ Human α2B Adrenergic Receptor Membrane Preparation
A
Adrenergic
alpha2B
Chem-1
HTS104M
ChemiSCREEN™ Membrane Preparation Recombinant Human β1 Adrenoceptor Receptor
A
Adrenergic
beta 1
Chem-1
HTS073M
ChemiScreen™ Recombinant Human β2 Adrenoceptor
A
Adrenergic
beta 2
Chem-2
HTS159M
ChemiSCREEN™ Membrane Preparation Recombinant Human β3 Adrenoceptor
A
Adrenergic
beta 3
Chem-1
HTS016M
ChemiSCREEN™ C3aR Membrane Preparation
A
Anaphylotoxin
C3aR
Chem-2
HTS017M
ChemiSCREEN™ C5aR Membrane Preparation, recombinant
A
Anaphylotoxin
C5aR
Chem-1
HTS064M
ChemiSCREEN™ Human Angiotensin II Receptor, Type I Membrane Preparation
A
Angiotensin
AT1
Chem-1
HTS208M
ChemiSCREEN™ Membrane Preparation Recombinant Human AT2 Angiotensin II Receptor
A
Angiotensin
AT2
Chem-1
HTS068M
ChemiSCREEN™ Membrane Preparation Recombinant Human APJ Apelin Receptor
A
Apelin
APJ
Chem-1
HTS123M
ChemiScreen™ Recombinant Human BB1 Bombesin/Neuromedin B Receptor Membrane Preparation
A
Bombesin
BB1
Chem-1
HTS084M
ChemiScreen™ BB2 Bombesin Receptor Membrane Preparation
A
Bombesin
BB2
Chem-1
HTS160M
ChemiSCREEN™ Membrane Preparation Recombinant Human BB3 Bombesin Receptor
A
Bombesin
BB3
Chem-1
HTS041M
ChemiScreen™ Bradykinin B2 Membrane Preparation
A
Bradykinin
B2
Chem-1
HTS127M
ChemiScreen™ Membrane Preparation Recombinant Human AMY1 Calcitonin Receptor
B
Calcitonin
AMY1
Chem-1
HTS172M
ChemiScreen™Human CGRP1 Calcitonin Receptor Membrane Preparation
B
Calcitonin
CGRP1
Chem-1
HTS019M
ChemiSCREEN™ CB1 Membrane Preparation
A
Cannabinoid
CB1
Chem-1
HTS020M
ChemiSCREEN™ Membrane Preparation Recombinant Human CB2 Cannabinoid Receptor
A
Cannabinoid
CB2
CHO (Chinese hamster ovary cells)
HTS020M2
ChemiSCREEN™ Membrane Preparation Recombinant Human CB2 Canabinoid Receptor Optimized for GTPγS Assay
A
Cannabinoid
CB2
Chem-4
HTS071M
ChemiSCREEN™ Membrane Preparation Recombinant Human ChemR23 Chemoattractant Receptor
A
Chemoattractant
ChemR23 / CMKLR1
Chem-1
HTS005M
ChemiSCREEN™ CCR1 Membrane Preparation
A
Chemokine
CCR1
Chem-2
HTS014M
ChemiSCREEN™ CCR10 Membrane Preparation
A
Chemokine
CCR10
Chem-1
HTS007M
ChemiSCREEN™ CCR2B Membrane Preparation
A
Chemokine
CCR2B
Chem-1
HTS008M
ChemiSCREEN™ Membrane Preparation Recombinant Human CCR3 Chemokine Receptor
A
Chemokine
CCR3
Chem-1
HTS009M
ChemiSCREEN™ Membrane Preparation Recombinant Human CCR4 Chemokine Receptor
A
Chemokine
CCR4
Chem-1
HTS010M
ChemiSCREEN™ Membrane Preparation Recombinant Rehsus Macaque CCR5 Chemokine Receptor
A
Chemokine
CCR5
Chem-1
HTS011M
ChemiSCREEN™ CCR6 Membrane Preparation
A
Chemokine
CCR6
Chem-1
HTS012M
ChemiSCREEN™ CCR7 Membrane Preparation, recombinant
A
Chemokine
CCR7
Chem-2
HTS013M
ChemiSCREEN™ CCR8 Membrane Preparation
A
Chemokine
CCR8
Chem-1
HTS036M
ChemiSCREEN™ CCR9 Membrane Preparation
A
Chemokine
CCR9
Chem-1
HTS015M
ChemiSCREEN™ CX3CR1 Membrane Preparation
A
Chemokine
CX3CR1
Chem-1
HTS001M
ChemiSCREEN™ Membrane Preparation Recombinant Human CXCR1 Chemokine Receptor
A
Chemokine
CXCR1 / IL-8a
Chem-1
HTS002M
ChemiScreen™ CXCR2 Membrane Preparation
A
Chemokine
CXCR2 / IL-8b
Chem-1
HTS003M
ChemiSCREEN™ Membrane Preparation Recombinant Human CXCR3 Chemokine Receptor
A
Chemokine
CXCR3
Chem-1
HTS004M
ChemiSCREEN™ CXCR4 Membrane Preparation
A
Chemokine
CXCR4
Chem-1
HTS055M
ChemiSCREEN™ Membrane Preparation Recombinant Human CXCR5 Chemokine Receptor
A
Chemokine
CXCR5
Chem-5
HTS054M
ChemiScreen™ CXCR6 Membrane Preparation
A
Chemokine
CXCR6
Chem-5
HTS138M
ChemiSCREEN™ Membrane Preparation Recombinant Human CXCR7 Chemokine Receptor
A
Chemokine
CXCR7 / RDC1
Chem-1
HTS184M
ChemiSCREEN™ Membrane Preparation Recombinant Human CCK1 Cholecystokinin Receptor
A
Cholecystokinin
CCK1 / CCKa
Chem-1
HTS083M
ChemiScreen™ Recombinant Human CCK2 Cholecystokinin Receptor Membrane Preparation
A
Cholecystokinin
CCK2 / CCKb
Chem-1
HTS000MC
ChemiSCREEN™ CHO Membrane Preparation, Null Control
Control
CHO (Chinese hamster ovary cells)
HTS000MC1
ChemiSCREEN™ Chem-1 Membrane Preparation, Null Control
Control
Chem-1
HTS000MC2
ChemiSCREEN™ Chem-2 Membrane Preparation, Null Control
Control
Chem-2
HTS023M
ChemiSCREEN™ CRF1 Membrane Preparation
B
CRF Receptor
CRF1
Chem-1
HTS024M
ChemiSCREEN™ Membrane Preparation Recombinant Human CRF2 Neuropeptide Receptor
B
CRF Receptor
CRF2
Chem-1
HTS102M
ChemiScreen™ D1 Dopamine Receptor Membrane Preparation
A
Dopamine
D1
Chem-1
HTS039M
ChemiSCREEN™ Membrane Preparation Recombinant Human D2 Dopamine Receptor
A
Dopamine
D2L
Chem-1
HTS103M
ChemiSCREEN™ Human D3 Dopamine Receptor Membrane Preparation
A
Dopamine
D3
Chem-1
HTS223M
ChemiSCREEN™ Membrane Preparation Recombinant Human D4 Dopamine Receptor
A
Dopamine
D4
Chem-1
HTS129M
ChemiScreen™ D5 Dopamine Receptor Membrane Preparation
A
Dopamine
D5
Chem-1
HTS070M
ChemiScreen™ Membrane Preparation Recombinant Human ETA Endothelin Receptor, Type A
A
Endothelin
ETA
Chem-1
HTS046M
ChemiSCREEN™ Membrane Preparation Recombinant Human ETB Endothelin Receptor
A
Endothelin
ETB
CHO (Chinese hamster ovary cells)
HTS063M
ChemiSCREEN™ Membrane Preparation Recombinant Human GPR43 Free Fatty Acid Receptor
A
Free Fatty Acid
FFA2 / GPR43
Chem-1
HTS135M
ChemiSCREEN™ Membrane Preparation Recombinant Human GPR41 Free Fatty Acid Receptor
A
Free Fatty Acid
FFA3 / GPR41
Chem-2
HTS119M
ChemiSCREEN™ Membrane Preparation Recombinant Human GABAB1b /GABAB2 Receptor
C
GABAB
GABAB1b
Chem-1
HTS094M
ChemiSCREEN™ Membrane Preparation Recombinant Human GAL1 Receptor
A
Galanin
GAL1
Chem-1
HTS186M
ChemiSCREEN™ Membrane Preparation Recombinant Human GAL2 Galanin Receptor
A
Galanin
GAL2
Chem-1
HTS187M
ChemiSCREEN™ Membrane Preparation Recombinant Human Gherlin Receptor
A
Ghrelin
Ghrelin / GHSR-1a / growth hormone secretagogue receptor
Chem-1
HTS134M
ChemiSCREEN™ Membrane Preparation Recombinant Human GIP Glucagon Family Receptor
B
Glucagon
GIP
Chem-9
HTS163M
ChemiSCREEN™ Membrane Preparation Recombinant Human GLP-1
B
Glucagon
GLP-1
Chem-9
HTS112M
ChemiScreen™ Recombinant Human Glucagon Receptor Membrane Preparation
B
Glucagon
glucagon / GCG
Chem-1
HTS146M
ChemiSCREEN™ Membrane Preparation Recombinant Human mGLU2 Metabotropic Glutamate Receptor
C
Glutamate (metabotropic)
mGlu2
Chem-1
HTS149M
ChemiSCREEN™ Membrane Preparation Recombinant Human mGlu6 Metabotropic Glutamate Receptor
C
Glutamate (metabotropic)
mGlu6
Chem-1
HTS027M
ChemiSCREEN™ GnRH Membrane Preparation
A
GnRH
GnRH / LHRH
Chem-1
HTS050M
ChemiScreen™ H1 Membrane Preparation
A
Histamine
H1
Chem-3
HTS086M
ChemiSCREEN™ Human H2 Histamine Receptor Membrane Preparation
A
Histamine
H2
Chem-2
HTS042M
ChemiScreen™ BLT1 Membrane Preparation
A
Leukotriene
BLT1
Chem-1
HTS061M
ChemiSCREEN™ Membrane Preparation Recombinant Human CysLT1 Cysteinyl Leukotriene Receptor
A
Leukotriene
CysLT1
Chem-1
HTS089M
ChemiSCREEN™ Membrane Preparation Recombinant Human LPA1 Lysophospholipid Receptor
A
Lysophospholipid
LPA1 / EDG2
Chem-1
HTS176M
ChemiSCREEN™ Membrane Preparation Recombinant Human S1P1 Lysophospholipid Receptor
A
Lysophospholipid
S1P1 / EDG1
Chem-1
HTS078M
ChemiSCREEN™ Human Recombinant S1P2 Lysophospholipid Receptor Membrane Preparation
A
Lysophospholipid
S1P2 / EDG5
Chem-1
HTS097M
ChemiSCREEN™ Membrane Preparation Recombinant Human S1P3 Lysophospholipid Receptor
A
Lysophospholipid
S1P3 / EDG3
Chem-1
HTS193M
ChemiSCREEN™ Membrane Preparation Recombinant Human S1P5 Lysophospholipid Receptor
A
Lysophospholipid
S1P5 / EDG8
Chem-5
HTS206M
ChemiSCREEN™ Membrane Preparation Recombinant Human MrgD Mas-Related Gene Family Receptor
A
Mas-related gene
MRGPRD / MrgD
Chem-1
HTS122M
ChemiSCREEN™ Membrane Preparation Recombinant Human MrgX1 Receptor
A
Mas-related gene
MRGX1 / MRGPRX1
Chem-1
HTS025M
ChemiSCREEN™ Membrane Preparation Recombinant Human MCH1 Receptor
A
Melanin-concentrating hormone
MCHR1 / GPR24
Chem-1
HTS156M
ChemiSCREEN™ Membrane Preparation Recombinant Human MC1 Melanocortin Receptor
A
Melanocortin
MC1
Chem-1
HTS022M
ChemiSCREEN™ MC3 Membrane Preparation
A
Melanocortin
MC3
Chem-1
HTS105M
ChemiSCREEN™ Human MC4 Melanocortin Receptor Membrane Preparation
A
Melanocortin
MC4
Chem-3
HTS155M
ChemiSCREEN™ Membrane Preparation Recombinant Human MC5 Melanocortin Receptor
A
Melanocortin
MC5
Chem-1
HTS065M
ChemiSCREEN™ Membrane Preparation Recombinant Human MT1 Melatonin Receptor
A
Melatonin
MT1
Chem-1
HTS106M
ChemiSCREEN™ Membrane Preparation Recombinant Human MT2 Melatonin Receptor
A
Melatonin
MT2
Chem-1
HTS121M
ChemiSCREEN™ Human Motilin Receptor Membrane Preparation
A
Motilin
motilin receptor / MTLR / GPR38
Chem-1
HTS062M
ChemiScreen™ Recombinant Human NMU1 Neuromedin Receptor
A
Neuromedin U
NMU1
Chem-1
HTS098M
ChemiSCREEN™ Membrane Preparation Recombinant Human NMU2 Neuromedin U Receptor
A
Neuromedin U
NMU2
Chem-1
HTS180M
ChemiSCREEN™ Membrane Preparation Recombinant Human NPBW1 Neuropeptide B/W Receptor
A
Neuropeptide B/W
NPBW1 / GPR7
Chem-1
HTS181M
ChemiSCREEN™ Membrane Preparation Recombinant Human NPBW2 Neuropeptide B/W Receptor
A
Neuropeptide B/W
NPBW2 / GPR8
Chem-1
HTS066M
ChemiSCREEN™ Human Y2 Neuropeptide Receptor Membrane Preparation
A
Neuropeptide Y
Y2
Chem-1
HTS204M
ChemiSCREEN™ Membrane Preparation Recombinant Human Y4 Neuropeptide Y Receptor
A
Neuropeptide Y
Y4
Chem-1
HTS034M
ChemiSCREEN™ NTR1 Membrane Preparation
A
Neurotensin
NTR1 / NTS1
Chem-2
HTS018M
ChemiSCREEN™ FPR1 Membrane Preparation
A
N-formylpeptide
FPR1
Chem-2
HTS056M
ChemiScreen™ Membrane Preparation Recombinant Human FPRL1 (Formyl Peptide Receptor-Like 1)
A
N-formylpeptide
FPRL1 / ALX / HM63
Chem-1
HTS201M
ChemiSCREEN™ Membrane Preparation Recombinant Human GPR109A Receptor
A
Nicotinic Acid
GPR109A
Chem-4
HTS100M
ChemiSCREEN™ Human δ Opioid Receptor Membrane Preparation
A
Opioid
Delta / OP1 / DOP / DOR
Chem-1
HTS095M
ChemiScreen™ Membrane Preparation Recombinant Human Kappa Opioid Receptor
A
Opioid
Kappa / OP2 / KOP / KOR
Chem-1
HTS101M
CHEMISCREEN™ MEMBRANE PREPARATION RECOMBINANT HUMAN µ (Mu) OPIOID RECEPTOR
A
Opioid
Mu / OP3 / MOP / MOR
Chem-5
HTS040M
ChemiSCREEN™ Membrane Preparation Recombinant Human NOP Opioid Receptor
A
Opioid
NOP / ORL1 / OP4
Chem-1
HTS090M
ChemiScreen™ Recombinant Human OT Oxytocin Receptor Membrane Preparation
A
Oxytocin
OT
Chem-1
HTS189M
ChemiSCREEN™ Membrane Preparation Recombinant Human GPR103 / QRFP Neuropeptide Receptor
A
Peptide P518
GPR103 / QRFP
Chem-1
HTS074M
ChemiSCREEN™ Human PK1 Prokineticin Receptor Membrane Preparation
A
Prokineticin
PK1 / PKR1
Chem-1
HTS182M
ChemiSCREEN™ Membrane Preparation Recombinant Human PK2 Prokineticin Receptor
A
Prokineticin
PK2 / PKR2
Chem-1
HTS057M
ChemiScreen™ Recombinant Human PRP/GPR10 Prolactin-Releasing Peptide Receptor Membrane Preparation
A
Prolactin-releasing peptide
PRP / PrRP / GPR10
Chem-1
HTS031M
ChemiSCREEN™ CRTH2 Membrane Preparation
A
Prostanoid
CRTH2 / DP2 / GPR44
Chem-1
HTS091M
ChemiSCREEN™ Human DP Prostanoid Receptor Membrane Preparation
A
Prostanoid
DP
Chem-1
HTS900PA
ChemiSCREEN™ Prostanoid Receptor Array Ready-to-Assay Plates Frozen Pre-Plated Membrane Preparation (96-well)
A
Prostanoid
DP2, DP, EP3, EP4, TP
Chem-1
HTS099M
ChemiSCREEN™ Membrane Preparation Recombinant Human EP1 Prostanoid Receptor
A
Prostanoid
EP1
Chem-1
HTS185M
ChemiSCREEN™ Membrane Preparation Recombinant Human EP2 Prostanoid Receptor
A
Prostanoid
EP2
Chem-1
HTS092M
ChemiSCREEN™ EP3 Prostanoid Receptor Membrane Preparation
A
Prostanoid
EP3
Chem-1
HTS142M
ChemiScreen™ Membrane Preparation Recombinant Human EP4 Prostanoid Receptor
A
Prostanoid
EP4
Chem-1
HTS142P
ChemiSCREEN™ EP4 Prostanoid Receptor Ready-to-Assay Plates Frozen Pre-Plated Membrane Preparation (96-well)
A
Prostanoid
EP4
Chem-1
HTS081M
ChemiScreen™ Membrane Preparation Recombinant Human TBXA2R (TP) Thromboxane Receptor
A
Prostanoid
TP / TXA2 / PGH2
Chem-1
HTS037M
ChemiSCREEN™ Membrane Preparation Recombinant Human PAR2 Protease-Activated Receptor
A
Protease-activated
PAR2
Chem-1
HTS030M
ChemiSCREEN™ PTH Membrane Preparation
B
PTH receptor
PTH1
Chem-1
HTS108M
ChemiSCREEN™ Membrane Preparation Recombinant Human 5-HT1B Serotonin Receptor
A
Serotonin
5-HT1B
Chem-1
HTS082M
ChemiSCREEN™ Human 5-HT2A Serotonin Receptor Membrane Preparation
A
Serotonin
5-HT2A
Chem-1
HTS132M
ChemiSCREEN™ Human 5-HT2C Receptor Membrane Preparation
A
Serotonin
5-HT2C
Chem-1
HTS110M
ChemiSCREEN™ Membrane Preparation Recombinant Human 5-HT4B Serotonin Receptor
A
Serotonin
5-HT4
Chem-1
HTS141M
ChemiSCREEN™ Membrane Preparation Recombinant Human 5-HT5A Serotonin Receptor
A
Serotonin
5-HT5A
Chem-1
HTS111M
ChemiSCREEN™ Membrane Preparation Recombinant Human 5-HT6 Serotonin Receptor
A
Serotonin
5-HT6
Chem-1
HTS215M
ChemiSCREEN™ Membrane Preparation Recombinant Human 5-HT₇ Serotonin Receptor
A
Serotonin
5-HT7
Chem-1
HTS170M
ChemiSCREEN™ Membrane Preparation Recombinant Human sst1 Somatostatin Receptor
A
Somatostatin
sst1
Chem-1
HTS028M
ChemiSCREEN™ Membrane Preparation Recombinant Human sst2 Somatostatin Receptor
A
Somatostatin
sst2
Chem-1
HTS125M
ChemiScreen™ Membrane Preparation Recombinant Human SST4 SOMATOSTATIN RECEPTOR
A
Somatostatin
sst4
Chem-1
HTS139M
ChemiSCREEN™ Membrane Preparation Recombinant Human sst5 Somatostatin Receptor
A
Somatostatin
sst5
Chem-1
HTS080M
ChemiSCREEN™ Human NK1 Tachykinin Receptor Membrane Preparation
A
Tackykinin /neurokinin
NK1
Chem-1
HTS144M
ChemiSCREEN™ Membrane Preparation Recombinant Human NK2 Tachykinin Receptor
A
Tackykinin /neurokinin
NK2
Chem-1
HTS033M
ChemiSCREEN™ GPR14 Membrane Preparation
A
Urotensin II
UT / UT1 / GPR14
Chem-2
HTS059M
ChemiScreen™ V1A Vasopressin Membrane Preparation
A
Vasopressin
V1A
Chem-1
HTS136M
ChemiScreen™ Membrane Preparation Recombinant Human V1B Vasopressin Receptor
A
Vasopressin
V1B
Chem-1
HTS060M
ChemiScreen™ Human V2 Vasopressin Receptor Membrane Preparation
A
Vasopressin
V2
Chem-1
HTS114M
ChemiSCREEN™ Human PAC1 -long Receptor Membrane Preparation
B
VIP/PACAP
PAC1 long isoform / PACAP
Chem-1
HTS043M
ChemiScreen™ VPAC1 Membrane Preparation
B
VIP/PACAP
VPAC1 / VIP1
Chem-1
HTS079M
ChemiSCREEN™ Human VPAC2 VIP Receptor Membrane Preparation
B
VIP/PACAP
VPAC2 / VIP2
Chem-1