Reference Data
Defining Selectivity Signatures of Small Molecule Inhibitors
Publications
The specifities of protein kinase inhibitors: an update
— Jenny Bain, Hilary Mclauchlan, Matthew Elliott, Philip Cohen
Specificity and mechanism of action of some commonly used protein kinase inhibitors
— Stephen P. Davies, Helen Reddy, Matilde Caivano, Philip Cohen
Mechanistic considerations in high-throughput screening
— Robert A. Copeland
Inhibition Data
Kinase Inhibition Profile — Staurosporine.
Graphic illustrates the effect of Staurosporine (1 μM) on a wide variety of protein kinases assayed at 10 μM ATP
